Explorer

Browse the GPCRome

398 receptors match — sorted by development interest.

Class
Development
System
Sort
GeneReceptorClassFamilyStructuresLigandsTDLDev. interest
PTGDRDP₁ receptorAProstanoid receptors—916Tclin
52
FFAR1FFA1 receptorAFree fatty acid receptors9907Tclin
52
MC5RMC₅ receptorAMelanocortin receptors2906Tclin
52
CCR6CCR6AChemokine receptors3669Tchem
52
F2RL1PAR2AProteinase-activated receptors3468Tchem
51
GPER1GPERAEstrogen (G protein-coupled) receptors5223Tclin
51
FFAR4FFA4 receptorAFree fatty acid receptors12905Tchem
51
CYSLTR2CysLT₂ receptorALeukotriene receptors4488Tclin
51
PTGDR2DP₂ receptorAProstanoid receptors6921Tclin
51
GRM2mGlu₂ receptorCMetabotropic glutamate receptors23923Tchem
51
CXCR3CXCR3AChemokine receptors6917Tchem
50
CCR3CCR3AChemokine receptors1923Tchem
50
FPR2FPR2/ALXAFormylpeptide receptors9942Tchem
50
RHORhodopsinAOpsins4—Tbio
50
NPY1RY₁ receptorANeuropeptide Y receptors6511Tchem
50
MC2RMC₂ receptorAMelanocortin receptors160Tclin
50
GRM3mGlu₃ receptorCMetabotropic glutamate receptors8445Tchem
50
CXCR1CXCR1AChemokine receptors1723Tclin
50
CCKBRCCK₂ receptorACholecystokinin receptors5913Tchem
49
GPR183GPR183◇AClass A orphans2277Tclin
49
P2RY2P2Y₂ receptorAP2Y receptors—723Tclin
49
GPBAR1GPBA receptorABile acid receptors5909Tclin
49
OPRL1NOP receptorAOpioid receptors4909Tchem
49
NTSR1NTS₁ receptorANeurotensin receptors8901Tchem
49
APLNRapelin receptorAApelin receptors14926Tchem
49
SSTR4SST4 receptorASomatostatin receptors2925Tchem
49
NPY2RY₂ receptorANeuropeptide Y receptors5916Tchem
48
MCHR1MCH₁ receptorAMelanin-concentrating hormone10924Tchem
48
GRM7mGlu₇ receptorCMetabotropic glutamate receptors1418Tchem
48
GLP2RGLP-2 receptorB1Glucagon receptor family1237Tclin
48
CCR9CCR9AChemokine receptors1636Tchem
48
GPR119GPR119AGPR18, GPR55 and GPR1197919Tchem
47
TAS2R14TAS2R14T2Taste 2 receptors15328Tclin
47
C3AR1C3a receptorAComplement peptide receptors9452Tclin
47
GPR17GPR17◇AClass A orphans1551Tclin
47
CCR8CCR8AChemokine receptors6488Tchem
46
TACR2NK₂ receptorATachykinin receptors1912Tchem
46
BDKRB1B₁ receptorABradykinin receptors1927Tclin
46
P2RY6P2Y₆ receptorAP2Y receptors—711Tclin
45
GHRHRGHRH receptorB1Glucagon receptor family38Tclin
45
GALR1GAL₁ receptorAGalanin receptors2257Tchem
45
F2RL3PAR4AProteinase-activated receptors—905Tchem
45
RXFP1RXFP1ARelaxin family peptide receptors1853Tchem
44
GPR65GPR65◇AClass A orphans—139Tclin
44
ADCYAP1R1PAC₁ receptorB1VIP and PACAP receptors5227Tchem
44
GPR88GPR88◇AClass A orphans2759Tchem
44
CMKLR1chemerin receptorAChemerin receptor2568Tchem
43
GRM4mGlu₄ receptorCMetabotropic glutamate receptors4524Tchem
43
FFAR2FFA2 receptorAFree fatty acid receptors5907Tchem
43
GRPRBB₂ receptorABombesin receptors4481Tchem
43
FPR3FPR3AFormylpeptide receptors—812Tclin
43
GPR84GPR84◇AClass A orphans4909Tchem
43
VIPR2VPAC₂ receptorB1VIP and PACAP receptors2186Tchem
43
TRHRTRH₁ receptorAThyrotropin-releasing hormone receptors426Tchem
42
NPY5RY₅ receptorANeuropeptide Y receptors—913Tchem
42
GPR139GPR139◇AClass A orphans4699Tchem
42
SCTRsecretin receptorB1Glucagon receptor family327Tclin
42
LTB4RBLT₁ receptorALeukotriene receptors2796Tchem
42
CCR7CCR7AChemokine receptors146Tchem
42
BRS3BB₃ receptorABombesin receptors2352Tchem
42
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