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Browse the GPCRome
398 receptors match — sorted by development interest.
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| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| PTGDR | DP₁ receptor | A | Prostanoid receptors | — | 916 | Tclin | 52 |
| FFAR1 | FFA1 receptor | A | Free fatty acid receptors | 9 | 907 | Tclin | 52 |
| MC5R | MC₅ receptor | A | Melanocortin receptors | 2 | 906 | Tclin | 52 |
| CCR6 | CCR6 | A | Chemokine receptors | 3 | 669 | Tchem | 52 |
| F2RL1 | PAR2 | A | Proteinase-activated receptors | 3 | 468 | Tchem | 51 |
| GPER1 | GPER | A | Estrogen (G protein-coupled) receptors | 5 | 223 | Tclin | 51 |
| FFAR4 | FFA4 receptor | A | Free fatty acid receptors | 12 | 905 | Tchem | 51 |
| CYSLTR2 | CysLT₂ receptor | A | Leukotriene receptors | 4 | 488 | Tclin | 51 |
| PTGDR2 | DP₂ receptor | A | Prostanoid receptors | 6 | 921 | Tclin | 51 |
| GRM2 | mGlu₂ receptor | C | Metabotropic glutamate receptors | 23 | 923 | Tchem | 51 |
| CXCR3 | CXCR3 | A | Chemokine receptors | 6 | 917 | Tchem | 50 |
| CCR3 | CCR3 | A | Chemokine receptors | 1 | 923 | Tchem | 50 |
| FPR2 | FPR2/ALX | A | Formylpeptide receptors | 9 | 942 | Tchem | 50 |
| RHO | Rhodopsin | A | Opsins | 4 | — | Tbio | 50 |
| NPY1R | Y₁ receptor | A | Neuropeptide Y receptors | 6 | 511 | Tchem | 50 |
| MC2R | MC₂ receptor | A | Melanocortin receptors | 1 | 60 | Tclin | 50 |
| GRM3 | mGlu₃ receptor | C | Metabotropic glutamate receptors | 8 | 445 | Tchem | 50 |
| CXCR1 | CXCR1 | A | Chemokine receptors | 1 | 723 | Tclin | 50 |
| CCKBR | CCK₂ receptor | A | Cholecystokinin receptors | 5 | 913 | Tchem | 49 |
| GPR183 | GPR183◇ | A | Class A orphans | 2 | 277 | Tclin | 49 |
| P2RY2 | P2Y₂ receptor | A | P2Y receptors | — | 723 | Tclin | 49 |
| GPBAR1 | GPBA receptor | A | Bile acid receptors | 5 | 909 | Tclin | 49 |
| OPRL1 | NOP receptor | A | Opioid receptors | 4 | 909 | Tchem | 49 |
| NTSR1 | NTS₁ receptor | A | Neurotensin receptors | 8 | 901 | Tchem | 49 |
| APLNR | apelin receptor | A | Apelin receptors | 14 | 926 | Tchem | 49 |
| SSTR4 | SST4 receptor | A | Somatostatin receptors | 2 | 925 | Tchem | 49 |
| NPY2R | Y₂ receptor | A | Neuropeptide Y receptors | 5 | 916 | Tchem | 48 |
| MCHR1 | MCH₁ receptor | A | Melanin-concentrating hormone | 10 | 924 | Tchem | 48 |
| GRM7 | mGlu₇ receptor | C | Metabotropic glutamate receptors | 1 | 418 | Tchem | 48 |
| GLP2R | GLP-2 receptor | B1 | Glucagon receptor family | 1 | 237 | Tclin | 48 |
| CCR9 | CCR9 | A | Chemokine receptors | 1 | 636 | Tchem | 48 |
| GPR119 | GPR119 | A | GPR18, GPR55 and GPR119 | 7 | 919 | Tchem | 47 |
| TAS2R14 | TAS2R14 | T2 | Taste 2 receptors | 15 | 328 | Tclin | 47 |
| C3AR1 | C3a receptor | A | Complement peptide receptors | 9 | 452 | Tclin | 47 |
| GPR17 | GPR17◇ | A | Class A orphans | 1 | 551 | Tclin | 47 |
| CCR8 | CCR8 | A | Chemokine receptors | 6 | 488 | Tchem | 46 |
| TACR2 | NK₂ receptor | A | Tachykinin receptors | 1 | 912 | Tchem | 46 |
| BDKRB1 | B₁ receptor | A | Bradykinin receptors | 1 | 927 | Tclin | 46 |
| P2RY6 | P2Y₆ receptor | A | P2Y receptors | — | 711 | Tclin | 45 |
| GHRHR | GHRH receptor | B1 | Glucagon receptor family | 3 | 8 | Tclin | 45 |
| GALR1 | GAL₁ receptor | A | Galanin receptors | 2 | 257 | Tchem | 45 |
| F2RL3 | PAR4 | A | Proteinase-activated receptors | — | 905 | Tchem | 45 |
| RXFP1 | RXFP1 | A | Relaxin family peptide receptors | 1 | 853 | Tchem | 44 |
| GPR65 | GPR65◇ | A | Class A orphans | — | 139 | Tclin | 44 |
| ADCYAP1R1 | PAC₁ receptor | B1 | VIP and PACAP receptors | 5 | 227 | Tchem | 44 |
| GPR88 | GPR88◇ | A | Class A orphans | 2 | 759 | Tchem | 44 |
| CMKLR1 | chemerin receptor | A | Chemerin receptor | 2 | 568 | Tchem | 43 |
| GRM4 | mGlu₄ receptor | C | Metabotropic glutamate receptors | 4 | 524 | Tchem | 43 |
| FFAR2 | FFA2 receptor | A | Free fatty acid receptors | 5 | 907 | Tchem | 43 |
| GRPR | BB₂ receptor | A | Bombesin receptors | 4 | 481 | Tchem | 43 |
| FPR3 | FPR3 | A | Formylpeptide receptors | — | 812 | Tclin | 43 |
| GPR84 | GPR84◇ | A | Class A orphans | 4 | 909 | Tchem | 43 |
| VIPR2 | VPAC₂ receptor | B1 | VIP and PACAP receptors | 2 | 186 | Tchem | 43 |
| TRHR | TRH₁ receptor | A | Thyrotropin-releasing hormone receptors | 4 | 26 | Tchem | 42 |
| NPY5R | Y₅ receptor | A | Neuropeptide Y receptors | — | 913 | Tchem | 42 |
| GPR139 | GPR139◇ | A | Class A orphans | 4 | 699 | Tchem | 42 |
| SCTR | secretin receptor | B1 | Glucagon receptor family | 3 | 27 | Tclin | 42 |
| LTB4R | BLT₁ receptor | A | Leukotriene receptors | 2 | 796 | Tchem | 42 |
| CCR7 | CCR7 | A | Chemokine receptors | 1 | 46 | Tchem | 42 |
| BRS3 | BB₃ receptor | A | Bombesin receptors | 2 | 352 | Tchem | 42 |