Explorer
Browse the GPCRome
398 receptors match — sorted by development interest.
Class
Development
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| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| SSTR5 | SST5 receptor | A | Somatostatin receptors | 4 | 938 | Tclin | 63 |
| HTR5A | 5-HT5A receptor | A | 5-Hydroxytryptamine receptors | 5 | 753 | Tclin | 63 |
| MTNR1A | MT₁ receptor | A | Melatonin | 8 | 905 | Tclin | 62 |
| HCRTR2 | OX₂ receptor | A | Orexin receptors | 11 | 924 | Tclin | 62 |
| OXTR | OT receptor | A | Vasopressin and oxytocin receptors | 3 | 539 | Tclin | 62 |
| CCR2 | CCR2 | A | Chemokine receptors | 4 | 915 | Tclin | 62 |
| GABBR1 | GABAB1 | C | GABAB receptors | 1 | 224 | Tclin | 62 |
| PTGER2 | EP₂ receptor | A | Prostanoid receptors | 3 | 912 | Tclin | 61 |
| BDKRB2 | B₂ receptor | A | Bradykinin receptors | 3 | 910 | Tclin | 61 |
| AGTR2 | AT₂ receptor | A | Angiotensin receptors | 7 | 898 | Tclin | 61 |
| ADORA2B | A2B receptor | A | Adenosine receptors | 4 | 961 | Tclin | 61 |
| CCKAR | CCK₁ receptor | A | Cholecystokinin receptors | 12 | 880 | Tclin | 61 |
| PTGER4 | EP₄ receptor | A | Prostanoid receptors | 8 | 924 | Tclin | 61 |
| MTNR1B | MT₂ receptor | A | Melatonin | 5 | 524 | Tclin | 61 |
| HRH3 | H₃ receptor | A | Histamine receptors | 7 | 925 | Tclin | 61 |
| ADORA3 | A₃ receptor | A | Adenosine receptors | 2 | 971 | Tclin | 61 |
| F2R | PAR1 | A | Proteinase-activated receptors | 3 | 899 | Tclin | 60 |
| ADRA1B | α1B-adrenoceptor | A | Adrenoceptors | 1 | 525 | Tclin | 60 |
| PTGER3 | EP₃ receptor | A | Prostanoid receptors | 4 | 919 | Tclin | 60 |
| S1PR3 | S1P₃ receptor | A | Lysophospholipid (S1P) receptors | 4 | 906 | Tclin | 60 |
| PTGIR | IP receptor | A | Prostanoid receptors | 2 | 798 | Tclin | 60 |
| CALCR | CT receptor | B1 | Calcitonin receptors | 17 | 379 | Tclin | 60 |
| AVPR1A | V1A receptor | A | Vasopressin and oxytocin receptors | — | 938 | Tclin | 60 |
| CYSLTR1 | CysLT₁ receptor | A | Leukotriene receptors | 2 | 641 | Tclin | 59 |
| SSTR3 | SST3 receptor | A | Somatostatin receptors | 2 | 939 | Tclin | 59 |
| FPR1 | FPR1 | A | Formylpeptide receptors | 4 | 929 | Tclin | 59 |
| CX3CR1 | CX₃CR1 | A | Chemokine receptors | 2 | 405 | Tclin | 58 |
| HTR1E | 5-HT1E receptor | A | 5-Hydroxytryptamine receptors | 3 | 416 | Tclin | 58 |
| LPAR1 | LPA₁ receptor | A | Lysophospholipid (LPA) receptors | 16 | 915 | Tclin | 58 |
| TAAR1 | TA₁ receptor | A | Trace amine receptors | 17 | 506 | Tclin | 58 |
| SSTR1 | SST1 receptor | A | Somatostatin receptors | 2 | 922 | Tclin | 58 |
| TBXA2R | TP receptor | A | Prostanoid receptors | 4 | 921 | Tclin | 58 |
| S1PR5 | S1P₅ receptor | A | Lysophospholipid (S1P) receptors | 2 | 894 | Tclin | 58 |
| TACR3 | NK₃ receptor | A | Tachykinin receptors | 3 | 898 | Tclin | 58 |
| HRH4 | H₄ receptor | A | Histamine receptors | 10 | 908 | Tclin | 57 |
| MLNR | motilin receptor | A | Motilin receptors | 2 | 747 | Tclin | 57 |
| FSHR | FSH receptor | A | Glycoprotein hormone receptors | 2 | 221 | Tclin | 57 |
| CNR2 | CB₂ receptor | A | Cannabinoid receptors | 9 | 924 | Tclin | 57 |
| MRGPRX2 | MRGPRX2◇ | A | Class A orphans | 14 | 282 | Tclin | 57 |
| C5AR1 | C5a₁ receptor | A | Complement peptide receptors | 10 | 921 | Tclin | 57 |
| GPR35 | GPR35◇ | A | Class A orphans | 1 | 784 | Tclin | 57 |
| LHCGR | LH receptor | A | Glycoprotein hormone receptors | 4 | 137 | Tclin | 57 |
| HTR1F | 5-HT1F receptor | A | 5-Hydroxytryptamine receptors | 1 | 322 | Tclin | 56 |
| AVPR1B | V1B receptor | A | Vasopressin and oxytocin receptors | — | 926 | Tclin | 56 |
| KISS1R | kisspeptin receptor | A | Kisspeptin receptors | 5 | 629 | Tchem | 55 |
| GPR55 | GPR55 | A | GPR18, GPR55 and GPR119 | 4 | 820 | Tclin | 55 |
| PTAFR | PAF receptor | A | Platelet-activating factor receptors | 3 | 836 | Tclin | 55 |
| CXCR2 | CXCR2 | A | Chemokine receptors | 3 | 908 | Tchem | 55 |
| GABBR2 | GABAB2 | C | GABAB receptors | 12 | 182 | Tclin | 55 |
| GRM5 | mGlu₅ receptor | C | Metabotropic glutamate receptors | 21 | 919 | Tchem | 55 |
| PTGER1 | EP₁ receptor | A | Prostanoid receptors | — | 917 | Tclin | 54 |
| CCR4 | CCR4 | A | Chemokine receptors | — | 906 | Tclin | 54 |
| CCR1 | CCR1 | A | Chemokine receptors | 3 | 916 | Tchem | 54 |
| MC3R | MC₃ receptor | A | Melanocortin receptors | 1 | 907 | Tclin | 54 |
| HCAR2 | HCA₂ receptor | A | Hydroxycarboxylic acid receptors | 34 | 894 | Tclin | 53 |
| GRM1 | mGlu₁ receptor | C | Metabotropic glutamate receptors | 3 | 895 | Tchem | 53 |
| ACKR3 | ACKR3 | A | Chemokine receptors | 7 | 903 | Tclin | 53 |
| S1PR4 | S1P₄ receptor | A | Lysophospholipid (S1P) receptors | — | 896 | Tclin | 53 |
| S1PR2 | S1P₂ receptor | A | Lysophospholipid (S1P) receptors | 1 | 866 | Tclin | 53 |
| P2RY1 | P2Y₁ receptor | A | P2Y receptors | 4 | 920 | Tclin | 52 |