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Browse the GPCRome

398 receptors match — sorted by development interest.

Class
Development
System
Sort
GeneReceptorClassFamilyStructuresLigandsTDLDev. interest
SSTR5SST5 receptorASomatostatin receptors4938Tclin
63
HTR5A5-HT5A receptorA5-Hydroxytryptamine receptors5753Tclin
63
MTNR1AMT₁ receptorAMelatonin8905Tclin
62
HCRTR2OX₂ receptorAOrexin receptors11924Tclin
62
OXTROT receptorAVasopressin and oxytocin receptors3539Tclin
62
CCR2CCR2AChemokine receptors4915Tclin
62
GABBR1GABAB1CGABAB receptors1224Tclin
62
PTGER2EP₂ receptorAProstanoid receptors3912Tclin
61
BDKRB2B₂ receptorABradykinin receptors3910Tclin
61
AGTR2AT₂ receptorAAngiotensin receptors7898Tclin
61
ADORA2BA2B receptorAAdenosine receptors4961Tclin
61
CCKARCCK₁ receptorACholecystokinin receptors12880Tclin
61
PTGER4EP₄ receptorAProstanoid receptors8924Tclin
61
MTNR1BMT₂ receptorAMelatonin5524Tclin
61
HRH3H₃ receptorAHistamine receptors7925Tclin
61
ADORA3A₃ receptorAAdenosine receptors2971Tclin
61
F2RPAR1AProteinase-activated receptors3899Tclin
60
ADRA1Bα1B-adrenoceptorAAdrenoceptors1525Tclin
60
PTGER3EP₃ receptorAProstanoid receptors4919Tclin
60
S1PR3S1P₃ receptorALysophospholipid (S1P) receptors4906Tclin
60
PTGIRIP receptorAProstanoid receptors2798Tclin
60
CALCRCT receptorB1Calcitonin receptors17379Tclin
60
AVPR1AV1A receptorAVasopressin and oxytocin receptors—938Tclin
60
CYSLTR1CysLT₁ receptorALeukotriene receptors2641Tclin
59
SSTR3SST3 receptorASomatostatin receptors2939Tclin
59
FPR1FPR1AFormylpeptide receptors4929Tclin
59
CX3CR1CX₃CR1AChemokine receptors2405Tclin
58
HTR1E5-HT1E receptorA5-Hydroxytryptamine receptors3416Tclin
58
LPAR1LPA₁ receptorALysophospholipid (LPA) receptors16915Tclin
58
TAAR1TA₁ receptorATrace amine receptors17506Tclin
58
SSTR1SST1 receptorASomatostatin receptors2922Tclin
58
TBXA2RTP receptorAProstanoid receptors4921Tclin
58
S1PR5S1P₅ receptorALysophospholipid (S1P) receptors2894Tclin
58
TACR3NK₃ receptorATachykinin receptors3898Tclin
58
HRH4H₄ receptorAHistamine receptors10908Tclin
57
MLNRmotilin receptorAMotilin receptors2747Tclin
57
FSHRFSH receptorAGlycoprotein hormone receptors2221Tclin
57
CNR2CB₂ receptorACannabinoid receptors9924Tclin
57
MRGPRX2MRGPRX2◇AClass A orphans14282Tclin
57
C5AR1C5a₁ receptorAComplement peptide receptors10921Tclin
57
GPR35GPR35◇AClass A orphans1784Tclin
57
LHCGRLH receptorAGlycoprotein hormone receptors4137Tclin
57
HTR1F5-HT1F receptorA5-Hydroxytryptamine receptors1322Tclin
56
AVPR1BV1B receptorAVasopressin and oxytocin receptors—926Tclin
56
KISS1Rkisspeptin receptorAKisspeptin receptors5629Tchem
55
GPR55GPR55AGPR18, GPR55 and GPR1194820Tclin
55
PTAFRPAF receptorAPlatelet-activating factor receptors3836Tclin
55
CXCR2CXCR2AChemokine receptors3908Tchem
55
GABBR2GABAB2CGABAB receptors12182Tclin
55
GRM5mGlu₅ receptorCMetabotropic glutamate receptors21919Tchem
55
PTGER1EP₁ receptorAProstanoid receptors—917Tclin
54
CCR4CCR4AChemokine receptors—906Tclin
54
CCR1CCR1AChemokine receptors3916Tchem
54
MC3RMC₃ receptorAMelanocortin receptors1907Tclin
54
HCAR2HCA₂ receptorAHydroxycarboxylic acid receptors34894Tclin
53
GRM1mGlu₁ receptorCMetabotropic glutamate receptors3895Tchem
53
ACKR3ACKR3AChemokine receptors7903Tclin
53
S1PR4S1P₄ receptorALysophospholipid (S1P) receptors—896Tclin
53
S1PR2S1P₂ receptorALysophospholipid (S1P) receptors1866Tclin
53
P2RY1P2Y₁ receptorAP2Y receptors4920Tclin
52
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