Explorer
Browse the GPCRome
398 receptors match — sorted by development interest.
Class
Development
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| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| GPR68 | GPR68◇ | A | Class A orphans | — | 79 | Tclin | 41 |
| NMUR2 | NMU2 receptor | A | Neuromedin U receptors | 3 | 275 | Tchem | 41 |
| GPR18 | GPR18 | A | GPR18, GPR55 and GPR119 | — | 305 | Tclin | 41 |
| PROKR1 | PKR₁ | A | Prokineticin receptors | — | 655 | Tchem | 41 |
| FZD7 | FZD₇ | F | Frizzled | 4 | 75 | Tchem | 41 |
| TAS2R38 | TAS2R38 | T2 | Taste 2 receptors | — | 22 | Tclin | 41 |
| GRM6 | mGlu₆ receptor | C | Metabotropic glutamate receptors | — | 242 | Tchem | 40 |
| SUCNR1 | succinate receptor | A | Succinate receptors | 7 | 204 | Tchem | 40 |
| PROKR2 | PKR₂ | A | Prokineticin receptors | — | 23 | Tchem | 40 |
| NPSR1 | NPS receptor | A | Neuropeptide S receptors | — | 592 | Tchem | 40 |
| GPR6 | GPR6◇ | A | Class A orphans | 4 | 501 | Tchem | 39 |
| GPR52 | GPR52◇ | A | Class A orphans | 5 | 763 | Tchem | 39 |
| P2RY4 | P2Y₄ receptor | A | P2Y receptors | — | 413 | Tclin | 39 |
| FZD4 | FZD₄ | F | Frizzled | 3 | 3 | Tchem | 39 |
| GALR2 | GAL₂ receptor | A | Galanin receptors | 4 | 288 | Tchem | 39 |
| MRGPRX1 | MRGPRX1◇ | A | Class A orphans | 7 | 311 | Tclin | 38 |
| LGR4 | LGR4◇ | A | Class A orphans | 9 | 6 | Tchem | 38 |
| CCRL2 | CCRL2 | A | Chemokine receptors | — | 307 | Tchem | 38 |
| NMUR1 | NMU1 receptor | A | Neuromedin U receptors | 2 | 255 | Tchem | 38 |
| CXCR5 | CXCR5 | A | Chemokine receptors | — | 155 | Tchem | 38 |
| LTB4R2 | BLT₂ receptor | A | Leukotriene receptors | — | 498 | Tclin | 38 |
| NMBR | BB₁ receptor | A | Bombesin receptors | 1 | 312 | Tchem | 37 |
| HCAR3 | HCA₃ receptor | A | Hydroxycarboxylic acid receptors | 4 | 239 | Tchem | 37 |
| VIPR1 | VPAC₁ receptor | B1 | VIP and PACAP receptors | 3 | 100 | Tchem | 37 |
| GPR39 | GPR39◇ | A | Class A orphans | — | 166 | Tchem | 37 |
| GRM8 | mGlu₈ receptor | C | Metabotropic glutamate receptors | — | 293 | Tchem | 37 |
| P2RY14 | P2Y₁₄ receptor | A | P2Y receptors | — | 733 | Tchem | 37 |
| GPR174 | GPR174◇ | A | Class A orphans | 3 | 182 | Tchem | 37 |
| TAS1R3 | TAS1R3 | C | Taste 1 receptors | — | 377 | Tchem | 37 |
| LPAR3 | LPA₃ receptor | A | Lysophospholipid (LPA) receptors | — | 390 | Tchem | 37 |
| MCHR2 | MCH₂ receptor | A | Melanin-concentrating hormone | 1 | 257 | Tchem | 37 |
| RXFP4 | RXFP4 | A | Relaxin family peptide receptors | 3 | 144 | Tchem | 36 |
| NTSR2 | NTS₂ receptor | A | Neurotensin receptors | — | 361 | Tclin | 36 |
| PRLHR | PrRP receptor | A | Prolactin-releasing peptide receptors | 2 | 259 | Tchem | 36 |
| ADGRF1 | ADGRF1 | B2 | ADGRF | 9 | 34 | Tclin | 36 |
| FZD6 | FZD₆ | F | Frizzled | 2 | 4 | Tbio | 36 |
| HCAR1 | HCA₁ receptor | A | Hydroxycarboxylic acid receptors | — | 385 | Tclin | 35 |
| FFAR3 | FFA3 receptor | A | Free fatty acid receptors | 2 | 157 | Tchem | 35 |
| GPR4 | GPR4◇ | A | Class A orphans | — | 145 | Tchem | 35 |
| LPAR2 | LPA₂ receptor | A | Lysophospholipid (LPA) receptors | — | 397 | Tchem | 35 |
| LPAR6 | LPA₆ receptor | A | Lysophospholipid (LPA) receptors | — | 23 | Tchem | 35 |
| RXFP3 | RXFP3 | A | Relaxin family peptide receptors | — | 274 | Tchem | 35 |
| NPY4R | Y₄ receptor | A | Neuropeptide Y receptors | 1 | 543 | Tchem | 35 |
| CRHR1 | CRF₁ receptor | B1 | Corticotropin-releasing factor receptors | 7 | — | Tbio | 35 |
| GPR132 | GPR132◇ | A | Class A orphans | 4 | 71 | Tchem | 35 |
| GPR143 | GPR143◇ | Other | Other GPCR orphans | — | 2 | Tclin | 35 |
| QRFPR | QRFP receptor | A | Peptide P518 receptors | 2 | 254 | Tchem | 35 |
| CXCR6 | CXCR6 | A | Chemokine receptors | — | 114 | Tchem | 34 |
| RXFP2 | RXFP2 | A | Relaxin family peptide receptors | — | 29 | Tchem | 34 |
| NPBWR1 | NPBW1 receptor | A | Neuropeptide W/neuropeptide B receptors | — | 550 | Tchem | 34 |
| NPFFR2 | NPFF2 receptor | A | Neuropeptide FF/neuropeptide AF receptors | — | 409 | Tchem | 34 |
| TAS1R2 | TAS1R2 | C | Taste 1 receptors | — | 180 | Tchem | 34 |
| MRGPRX4 | MRGPRX4◇ | A | Class A orphans | 4 | 513 | Tchem | 34 |
| FZD1 | FZD₁ | F | Frizzled | 2 | 11 | Tchem | 34 |
| GPRC5D | GPRC5D◇ | C | Class C Orphans | 2 | 1 | Tclin | 34 |
| P2RY11 | P2Y₁₁ receptor | A | P2Y receptors | — | 80 | Tclin | 34 |
| CCR10 | CCR10 | A | Chemokine receptors | — | 42 | Tchem | 33 |
| GPR3 | GPR3◇ | A | Class A orphans | 3 | 83 | Tchem | 33 |
| FZD2 | FZD₂ | F | Frizzled | — | 5 | Tchem | 33 |
| TAS2R46 | TAS2R46 | T2 | Taste 2 receptors | 3 | 39 | Tclin | 33 |