GPER1
ATclinGPER
Rhodopsin· Estrogen (G protein-coupled) receptors· 375 aa
Development interest
51/ 100
Tclin
An approved drug acts on this receptor.
1,853 refs·223 ligands·5 structures
Ligands
×20%
Literature
×30%
Structures
×15%
Approved drugs
×20%
Disease evidence
×15%
Signalling
Signal transduction
Primary G-protein coupling is not curated for GPER1 in Helix7. See GPCRdb couplings for transducer data on this receptor.
At a glance
Key facts
- Structures
- 5
- Distinct ligands
- 223
- Approved drugs
- 4
- Disease links
- 676
- Organ systems
- 11
- Citations
- 1,853
AdiposeCardiovascularDigestiveEndocrineImmuneIntegumentaryMusculoskeletalNervousReproductiveRespiratoryUrinary
Sources & attribution
GPCRdbCC BY 4.0Human Protein AtlasCC BY-SA 4.0IUPHAR/BPS Guide to PHARMACOLOGYCC BY-SA 4.0ChEMBLCC BY-SA 4.0PubChem BioAssayPublic domainOpen Targets PlatformCC0 1.0
Data redistributed under each source's licence. See Citation & licenses.