PTGER2

ATclin

EP2 receptor

Rhodopsin· Prostanoid receptors· 358 aa
Development interest
61/ 100
Tclin

An approved drug acts on this receptor.

759 refs·912 ligands·3 structures
Ligands
×20%
Disease evidence
×15%
Literature
×30%
Approved drugs
×20%
Structures
×15%
Signalling

Signal transduction

Primary G-protein transducer(s):

Gsprimary

Canonical coupling; some receptors also signal through secondary transducers and β-arrestin. See GPCRdb couplings for full data.

At a glance

Key facts

Structures
3
Distinct ligands
912
Approved drugs
8
Disease links
336
Organ systems
11
Citations
759
AdiposeCardiovascularDigestiveEndocrineImmuneIntegumentaryMusculoskeletalNervousReproductiveRespiratoryUrinary