Browse/Class A/ADORA2B

ADORA2B

ATclin

A2B receptor

Rhodopsin· Adenosine receptors· 332 aa
Development interest
61/ 100
Tclin

An approved drug acts on this receptor.

636 refs·961 ligands·4 structures
Ligands
×20%
Disease evidence
×15%
Literature
×30%
Approved drugs
×20%
Structures
×15%
Signalling

Signal transduction

Primary G-protein transducer(s):

Gsprimary

Canonical coupling; some receptors also signal through secondary transducers and β-arrestin. See GPCRdb couplings for full data.

At a glance

Key facts

Structures
4
Distinct ligands
961
Approved drugs
6
Disease links
519
Organ systems
10
Citations
636
CardiovascularDigestiveEndocrineImmuneIntegumentaryMusculoskeletalNervousReproductiveRespiratoryUrinary