PTGER4

ATclin

EP4 receptor

Rhodopsin· Prostanoid receptors· 488 aa
Development interest
61/ 100
Tclin

An approved drug acts on this receptor.

1,064 refs·924 ligands·8 structures
Ligands
×20%
Literature
×30%
Disease evidence
×15%
Structures
×15%
Approved drugs
×20%
Signalling

Signal transduction

Primary G-protein transducer(s):

Gsprimary

Canonical coupling; some receptors also signal through secondary transducers and β-arrestin. See GPCRdb couplings for full data.

At a glance

Key facts

Structures
8
Distinct ligands
924
Approved drugs
6
Disease links
979
Organ systems
11
Citations
1,064
AdiposeCardiovascularDigestiveEndocrineImmuneIntegumentaryMusculoskeletalNervousReproductiveRespiratoryUrinary