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Class A · Rhodopsin
287 receptors match — sorted by development interest.
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| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| ADRB2 | β₂-adrenoceptor | A | Adrenoceptors | 126 | 905 | Tclin | 84 |
| DRD2 | D₂ receptor | A | Dopamine receptors | 8 | 548 | Tclin | 82 |
| HTR2A | 5-HT2A receptor | A | 5-Hydroxytryptamine receptors | 18 | 974 | Tclin | 82 |
| OPRM1 | μ receptor | A | Opioid receptors | 10 | 953 | Tclin | 78 |
| HTR1A | 5-HT1A receptor | A | 5-Hydroxytryptamine receptors | 13 | 987 | Tclin | 78 |
| HRH1 | H₁ receptor | A | Histamine receptors | 7 | 558 | Tclin | 77 |
| DRD1 | D₁ receptor | A | Dopamine receptors | 22 | 418 | Tclin | 77 |
| HRH2 | H₂ receptor | A | Histamine receptors | 5 | 846 | Tclin | 77 |
| AGTR1 | AT₁ receptor | A | Angiotensin receptors | 9 | 904 | Tclin | 76 |
| DRD3 | D₃ receptor | A | Dopamine receptors | 6 | 923 | Tclin | 76 |
| CXCR4 | CXCR4 | A | Chemokine receptors | 14 | 918 | Tclin | 76 |
| EDNRB | ETB receptor | A | Endothelin receptors | 18 | 898 | Tclin | 75 |
| CHRM2 | M₂ receptor | A | Acetylcholine receptors (muscarinic) | 14 | 969 | Tclin | 75 |
| ADRB1 | β₁-adrenoceptor | A | Adrenoceptors | 4 | 904 | Tclin | 74 |
| CHRM1 | M₁ receptor | A | Acetylcholine receptors (muscarinic) | 6 | 951 | Tclin | 74 |
| ADRA2A | α2A-adrenoceptor | A | Adrenoceptors | 10 | 862 | Tclin | 74 |
| ADORA2A | A2A receptor | A | Adenosine receptors | 80 | 978 | Tclin | 74 |
| HTR2B | 5-HT2B receptor | A | 5-Hydroxytryptamine receptors | 11 | 903 | Tclin | 73 |
| OPRK1 | κ receptor | A | Opioid receptors | 11 | 938 | Tclin | 73 |
| CNR1 | CB₁ receptor | A | Cannabinoid receptors | 21 | 917 | Tclin | 73 |
| MC4R | MC₄ receptor | A | Melanocortin receptors | 11 | 906 | Tclin | 72 |
| HTR2C | 5-HT2C receptor | A | 5-Hydroxytryptamine receptors | 7 | 572 | Tclin | 72 |
| CHRM4 | M₄ receptor | A | Acetylcholine receptors (muscarinic) | 11 | 937 | Tclin | 72 |
| TSHR | TSH receptor | A | Glycoprotein hormone receptors | 7 | 584 | Tclin | 71 |
| DRD4 | D₄ receptor | A | Dopamine receptors | 3 | 904 | Tclin | 71 |
| HTR1B | 5-HT1B receptor | A | 5-Hydroxytryptamine receptors | 5 | 933 | Tclin | 71 |
| SSTR2 | SST2 receptor | A | Somatostatin receptors | 17 | 958 | Tclin | 70 |
| ADRA1A | α1A-adrenoceptor | A | Adrenoceptors | 6 | 910 | Tclin | 70 |
| CHRM3 | M₃ receptor | A | Acetylcholine receptors (muscarinic) | 4 | 582 | Tclin | 70 |
| EDNRA | ETA receptor | A | Endothelin receptors | 5 | 897 | Tclin | 70 |
| OPRD1 | δ receptor | A | Opioid receptors | 7 | 940 | Tclin | 69 |
| CCR5 | CCR5 | A | Chemokine receptors | 11 | 923 | Tclin | 69 |
| S1PR1 | S1P₁ receptor | A | Lysophospholipid (S1P) receptors | 17 | 921 | Tclin | 69 |
| AVPR2 | V₂ receptor | A | Vasopressin and oxytocin receptors | 5 | 936 | Tclin | 69 |
| ADORA1 | A₁ receptor | A | Adenosine receptors | 5 | 942 | Tclin | 69 |
| GNRHR | GnRH₁ receptor | A | Gonadotrophin-releasing hormone receptors | 1 | 923 | Tclin | 68 |
| MC1R | MC₁ receptor | A | Melanocortin receptors | 4 | 901 | Tclin | 67 |
| TACR1 | NK₁ receptor | A | Tachykinin receptors | 12 | 929 | Tclin | 67 |
| ADRA2C | α2C-adrenoceptor | A | Adrenoceptors | 1 | 873 | Tclin | 66 |
| ADRA2B | α2B-adrenoceptor | A | Adrenoceptors | 2 | 519 | Tclin | 66 |
| HTR7 | 5-HT₇ receptor | A | 5-Hydroxytryptamine receptors | 1 | 919 | Tclin | 65 |
| HTR1D | 5-HT1D receptor | A | 5-Hydroxytryptamine receptors | 1 | 955 | Tclin | 65 |
| HTR6 | 5-HT₆ receptor | A | 5-Hydroxytryptamine receptors | 3 | 942 | Tclin | 65 |
| P2RY12 | P2Y₁₂ receptor | A | P2Y receptors | 5 | 906 | Tclin | 65 |
| DRD5 | D₅ receptor | A | Dopamine receptors | 1 | 786 | Tclin | 65 |
| CHRM5 | M₅ receptor | A | Acetylcholine receptors (muscarinic) | 1 | 906 | Tclin | 64 |
| PTGFR | FP receptor | A | Prostanoid receptors | 8 | 915 | Tclin | 64 |
| HTR4 | 5-HT₄ receptor | A | 5-Hydroxytryptamine receptors | 3 | 902 | Tclin | 64 |
| ADRB3 | β₃-adrenoceptor | A | Adrenoceptors | 2 | 424 | Tclin | 64 |
| GHSR | ghrelin receptor | A | Ghrelin receptors | 7 | 916 | Tclin | 64 |
| ADRA1D | α1D-adrenoceptor | A | Adrenoceptors | — | 894 | Tclin | 63 |
| HCRTR1 | OX₁ receptor | A | Orexin receptors | 14 | 917 | Tclin | 63 |
| SSTR5 | SST5 receptor | A | Somatostatin receptors | 4 | 938 | Tclin | 63 |
| HTR5A | 5-HT5A receptor | A | 5-Hydroxytryptamine receptors | 5 | 753 | Tclin | 63 |
| MTNR1A | MT₁ receptor | A | Melatonin | 8 | 905 | Tclin | 62 |
| HCRTR2 | OX₂ receptor | A | Orexin receptors | 11 | 924 | Tclin | 62 |
| CCR2 | CCR2 | A | Chemokine receptors | 4 | 915 | Tclin | 62 |
| OXTR | OT receptor | A | Vasopressin and oxytocin receptors | 3 | 539 | Tclin | 62 |
| BDKRB2 | B₂ receptor | A | Bradykinin receptors | 3 | 910 | Tclin | 61 |
| PTGER2 | EP₂ receptor | A | Prostanoid receptors | 3 | 912 | Tclin | 61 |
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