CNR1

ATclin

CB1 receptor

Rhodopsin· Cannabinoid receptors· 472 aa
Development interest
73/ 100
Tclin

An approved drug acts on this receptor.

4,561 refs·917 ligands·21 structures
Ligands
×20%
Literature
×30%
Disease evidence
×15%
Structures
×15%
Approved drugs
×20%
Signalling

Signal transduction

Primary G-protein transducer(s):

Gi/Goprimary

Canonical coupling; some receptors also signal through secondary transducers and β-arrestin. See GPCRdb couplings for full data.

At a glance

Key facts

Structures
21
Distinct ligands
917
Approved drugs
8
Disease links
959
Organ systems
11
Citations
4,561
AdiposeCardiovascularDigestiveEndocrineImmuneIntegumentaryMusculoskeletalNervousReproductiveRespiratoryUrinary