Explorer

Tchem targets

120 receptors match — sorted by development interest.

Class
Development
System
Sort
GeneReceptorClassFamilyStructuresLigandsTDLDev. interest
KISS1Rkisspeptin receptorAKisspeptin receptors5629Tchem
55
CXCR2CXCR2AChemokine receptors3908Tchem
55
GRM5mGlu₅ receptorCMetabotropic glutamate receptors21919Tchem
55
CCR1CCR1AChemokine receptors3916Tchem
54
GRM1mGlu₁ receptorCMetabotropic glutamate receptors3895Tchem
53
CCR6CCR6AChemokine receptors3669Tchem
52
F2RL1PAR2AProteinase-activated receptors3468Tchem
51
FFAR4FFA4 receptorAFree fatty acid receptors12905Tchem
51
GRM2mGlu₂ receptorCMetabotropic glutamate receptors23923Tchem
51
CCR3CCR3AChemokine receptors1923Tchem
50
CXCR3CXCR3AChemokine receptors6917Tchem
50
FPR2FPR2/ALXAFormylpeptide receptors9942Tchem
50
NPY1RY₁ receptorANeuropeptide Y receptors6511Tchem
50
GRM3mGlu₃ receptorCMetabotropic glutamate receptors8445Tchem
50
CCKBRCCK₂ receptorACholecystokinin receptors5913Tchem
49
NTSR1NTS₁ receptorANeurotensin receptors8901Tchem
49
OPRL1NOP receptorAOpioid receptors4909Tchem
49
APLNRapelin receptorAApelin receptors14926Tchem
49
SSTR4SST4 receptorASomatostatin receptors2925Tchem
49
NPY2RY₂ receptorANeuropeptide Y receptors5916Tchem
48
MCHR1MCH₁ receptorAMelanin-concentrating hormone10924Tchem
48
GRM7mGlu₇ receptorCMetabotropic glutamate receptors1418Tchem
48
CCR9CCR9AChemokine receptors1636Tchem
48
GPR119GPR119AGPR18, GPR55 and GPR1197919Tchem
47
CCR8CCR8AChemokine receptors6488Tchem
46
TACR2NK₂ receptorATachykinin receptors1912Tchem
46
GALR1GAL₁ receptorAGalanin receptors2257Tchem
45
F2RL3PAR4AProteinase-activated receptors—905Tchem
45
RXFP1RXFP1ARelaxin family peptide receptors1853Tchem
44
ADCYAP1R1PAC₁ receptorB1VIP and PACAP receptors5227Tchem
44
GPR88GPR88◇AClass A orphans2759Tchem
44
CMKLR1chemerin receptorAChemerin receptor2568Tchem
43
GRM4mGlu₄ receptorCMetabotropic glutamate receptors4524Tchem
43
FFAR2FFA2 receptorAFree fatty acid receptors5907Tchem
43
GRPRBB₂ receptorABombesin receptors4481Tchem
43
GPR84GPR84◇AClass A orphans4909Tchem
43
VIPR2VPAC₂ receptorB1VIP and PACAP receptors2186Tchem
43
TRHRTRH₁ receptorAThyrotropin-releasing hormone receptors426Tchem
42
NPY5RY₅ receptorANeuropeptide Y receptors—913Tchem
42
GPR139GPR139◇AClass A orphans4699Tchem
42
BRS3BB₃ receptorABombesin receptors2352Tchem
42
CCR7CCR7AChemokine receptors146Tchem
42
LTB4RBLT₁ receptorALeukotriene receptors2796Tchem
42
NMUR2NMU2 receptorANeuromedin U receptors3275Tchem
41
PROKR1PKR₁AProkineticin receptors—655Tchem
41
FZD7FZD₇FFrizzled475Tchem
41
GRM6mGlu₆ receptorCMetabotropic glutamate receptors—242Tchem
40
SUCNR1succinate receptorASuccinate receptors7204Tchem
40
PROKR2PKR₂AProkineticin receptors—23Tchem
40
NPSR1NPS receptorANeuropeptide S receptors—592Tchem
40
GPR6GPR6◇AClass A orphans4501Tchem
39
GPR52GPR52◇AClass A orphans5763Tchem
39
FZD4FZD₄FFrizzled33Tchem
39
GALR2GAL₂ receptorAGalanin receptors4288Tchem
39
LGR4LGR4◇AClass A orphans96Tchem
38
CCRL2CCRL2AChemokine receptors—307Tchem
38
NMUR1NMU1 receptorANeuromedin U receptors2255Tchem
38
CXCR5CXCR5AChemokine receptors—155Tchem
38
NMBRBB₁ receptorABombesin receptors1312Tchem
37
HCAR3HCA₃ receptorAHydroxycarboxylic acid receptors4239Tchem
37
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