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Browse the GPCRome
398 receptors match — sorted by development interest.
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| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| UTS2R | UT receptor | A | Urotensin receptors | — | 520 | Tchem | 32 |
| TAS2R8 | TAS2R8 | T2 | Taste 2 receptors | — | 645 | Tclin | 32 |
| C5AR2 | C5a₂ receptor | A | Complement peptide receptors | — | 30 | Tclin | 32 |
| OXER1 | OXE receptor | A | Leukotriene receptors | — | 151 | Tchem | 32 |
| PTH2R | PTH2 receptor | B1 | Parathyroid hormone receptors | 1 | 25 | Tclin | 32 |
| GPR34 | GPR34◇ | A | Class A orphans | 9 | 37 | Tchem | 32 |
| LPAR5 | LPA₅ receptor | A | Lysophospholipid (LPA) receptors | — | 316 | Tchem | 32 |
| P2RY13 | P2Y₁₃ receptor | A | P2Y receptors | — | 35 | Tclin | 31 |
| LGR5 | LGR5◇ | A | Class A orphans | — | 5 | Tchem | 31 |
| GALR3 | GAL₃ receptor | A | Galanin receptors | — | 229 | Tchem | 31 |
| FZD5 | FZD₅ | F | Frizzled | 1 | 1 | Tchem | 31 |
| NPFFR1 | NPFF1 receptor | A | Neuropeptide FF/neuropeptide AF receptors | — | 187 | Tchem | 31 |
| TAS2R1 | TAS2R1 | T2 | Taste 2 receptors | — | 10 | Tclin | 31 |
| GPR142 | GPR142◇ | A | Class A orphans | — | 409 | Tchem | 30 |
| ADGRG1 | ADGRG1 | B2 | ADGRG | 1 | — | Tbio | 30 |
| XCR1 | XCR1 | A | Chemokine receptors | 1 | 3 | Tchem | 29 |
| P2RY10 | P2RY10◇ | A | Class A orphans | 1 | 122 | Tchem | 29 |
| TAS2R16 | TAS2R16 | T2 | Taste 2 receptors | — | 15 | Tclin | 29 |
| OXGR1 | oxoglutarate receptor | A | Oxoglutarate receptors | — | 12 | Tbio | 28 |
| LPAR4 | LPA₄ receptor | A | Lysophospholipid (LPA) receptors | — | 43 | Tchem | 28 |
| TAS1R1 | TAS1R1 | C | Taste 1 receptors | — | 200 | Tchem | 28 |
| MAS1 | MAS1◇ | A | Class A orphans | — | 11 | Tchem | 28 |
| GPR27 | GPR27◇ | A | Class A orphans | — | 114 | Tchem | 28 |
| LGR6 | LGR6◇ | A | Class A orphans | — | 8 | Tchem | 27 |
| GPR161 | GPR161◇ | A | Class A orphans | 2 | — | Tbio | 27 |
| CELSR1 | CELSR1 | B2 | ADGRC | — | — | Tbio | 27 |
| FZD8 | FZD₈ | F | Frizzled | — | 2 | Tclin | 27 |
| GPR160 | GPR160◇ | A | Class A orphans | — | 58 | Tchem | 27 |
| ADGRV1 | ADGRV1 | B2 | ADGRV | — | — | Tbio | 26 |
| GPR101 | GPR101◇ | A | Class A orphans | 3 | — | Tbio | 26 |
| GPRC6A | GPRC6 receptor◇ | C | Class C Orphans | — | 8 | Tbio | 26 |
| OPN1LW | OPN1LW | A | Opsins | 1 | — | Tbio | 25 |
| FZD3 | FZD₃ | F | Frizzled | 3 | — | Tbio | 25 |
| GPR179 | GPR179◇ | C | Class C Orphans | 1 | — | Tbio | 25 |
| ADGRG6 | ADGRG6 | B2 | ADGRG | — | — | Tbio | 24 |
| GPR158 | GPR158◇ | C | Class C Orphans | 5 | — | Tbio | 24 |
| GPR37 | GPR37◇ | A | Class A orphans | — | 2 | Tchem | 24 |
| TAS2R43 | TAS2R43 | T2 | Taste 2 receptors | — | 15 | Tclin | 24 |
| TAS2R4 | TAS2R4 | T2 | Taste 2 receptors | — | 8 | Tclin | 24 |
| OPN1MW | OPN1MW | A | Opsins | — | — | Tbio | 24 |
| F2RL2 | PAR3 | A | Proteinase-activated receptors | — | — | Tbio | 24 |
| GPR12 | GPR12◇ | A | Class A orphans | 1 | 2 | Tbio | 24 |
| ACKR1 | ACKR1 | A | Chemokine receptors | 1 | — | Tbio | 24 |
| CELSR2 | CELSR2 | B2 | ADGRC | — | — | Tbio | 24 |
| GPR50 | GPR50◇ | A | Class A orphans | — | 1 | Tchem | 23 |
| ACKR2 | ACKR2 | A | Chemokine receptors | — | 6 | Tbio | 23 |
| ADGRG2 | ADGRG2 | B2 | ADGRG | — | 1 | Tchem | 23 |
| OPN1SW | OPN1SW | A | Opsins | — | — | Tbio | 23 |
| TAS2R31 | TAS2R31 | T2 | Taste 2 receptors | — | 25 | Tclin | 23 |
| ADGRL3 | ADGRL3 | B2 | ADGRL | 2 | — | Tbio | 23 |
| P2RY8 | P2RY8◇ | A | Class A orphans | — | — | Tbio | 23 |
| ADGRD1 | ADGRD1 | B2 | ADGRD | 2 | — | Tbio | 23 |
| ADGRE5 | ADGRE5 | B2 | ADGRE | 6 | 2 | Tbio | 23 |
| GPR15 | GPR15◇ | A | Class A orphans | 1 | 4 | Tchem | 23 |
| TAS2R39 | TAS2R39 | T2 | Taste 2 receptors | — | 17 | Tclin | 23 |
| MRGPRD | MRGPRD◇ | A | Class A orphans | 6 | 1 | Tbio | 22 |
| TAS2R10 | TAS2R10 | T2 | Taste 2 receptors | — | 13 | Tclin | 22 |
| ADGRL1 | ADGRL1 | B2 | ADGRL | — | — | Tbio | 22 |
| TAS2R20 | TAS2R20 | T2 | Taste 2 receptors | — | 7 | Tclin | 22 |
| GPR156 | GPR156◇ | C | Class C Orphans | 5 | — | Tbio | 22 |