Explorer
Browse the GPCRome
398 receptors match — sorted by development interest.
Class
Development
System
Sort
| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| GPR61 | GPR61◇ | A | Class A orphans | 3 | 3 | Tchem | 22 |
| GPR75 | GPR75◇ | A | Class A orphans | — | 1 | Tchem | 22 |
| GPR87 | GPR87◇ | A | Class A orphans | — | 3 | Tchem | 22 |
| ADGRG3 | ADGRG3 | B2 | ADGRG | 2 | 1 | Tclin | 21 |
| ACKR4 | ACKR4 | A | Chemokine receptors | — | 3 | Tchem | 21 |
| TAS2R50 | TAS2R50 | T2 | Taste 2 receptors | — | 3 | Tclin | 21 |
| CMKLR2 | chemerin receptor 2 | A | Chemerin receptor | 2 | 18 | Tchem | 21 |
| OPN4 | OPN4 | A | Opsins | — | — | Tbio | 21 |
| TAS2R9 | TAS2R9 | T2 | Taste 2 receptors | — | 6 | Tclin | 21 |
| TAAR5 | TAAR5◇ | A | Class A orphans | — | 2 | Tbio | 21 |
| RRH | RRH | A | Opsins | — | — | Tbio | 21 |
| GPR20 | GPR20◇ | A | Class A orphans | 3 | — | Tbio | 20 |
| GPRC5A | GPRC5A◇ | C | Class C Orphans | — | — | Tbio | 20 |
| ADGRE2 | ADGRE2 | B2 | ADGRE | — | — | Tbio | 20 |
| GPRC5B | GPRC5B◇ | C | Class C Orphans | — | — | Tbio | 20 |
| GPR37L1 | GPR37L1◇ | A | Class A orphans | — | 2 | Tchem | 19 |
| GPR137 | GPR137◇ | Other | Other GPCR orphans | — | — | Tbio | 19 |
| TAS2R5 | TAS2R5 | T2 | Taste 2 receptors | — | 4 | Tclin | 19 |
| TAS2R7 | TAS2R7 | T2 | Taste 2 receptors | — | 4 | Tclin | 19 |
| CELSR3 | CELSR3 | B2 | ADGRC | — | — | Tbio | 19 |
| GPR19 | GPR19◇ | A | Class A orphans | — | 1 | Tchem | 19 |
| FZD10 | FZD₁₀ | F | Frizzled | — | — | Tbio | 18 |
| ADGRL2 | ADGRL2 | B2 | ADGRL | — | 1 | Tchem | 18 |
| OPN5 | OPN5 | A | Opsins | — | — | Tbio | 18 |
| ADGRL4 | ADGRL4 | B2 | ADGRL | — | — | Tbio | 18 |
| TAS2R13 | TAS2R13 | T2 | Taste 2 receptors | — | 4 | Tclin | 18 |
| TAS2R19 | TAS2R19 | T2 | Taste 2 receptors | — | 1 | Tclin | 18 |
| TAS2R3 | TAS2R3 | T2 | Taste 2 receptors | — | 2 | Tclin | 18 |
| NPBWR2 | NPBW2 receptor | A | Neuropeptide W/neuropeptide B receptors | — | 5 | Tchem | 18 |
| GPR26 | GPR26◇ | A | Class A orphans | — | — | Tbio | 18 |
| TAS2R40 | TAS2R40 | T2 | Taste 2 receptors | — | 5 | Tclin | 18 |
| OPN3 | OPN3 | A | Opsins | — | — | Tbio | 17 |
| GPR32 | GPR32◇ | A | Class A orphans | — | 4 | Tchem | 17 |
| ADGRB1 | ADGRB1 | B2 | ADGRB | — | 1 | Tbio | 17 |
| TAS2R42 | TAS2R42 | T2 | Taste 2 receptors | — | 1 | Tclin | 17 |
| GPR135 | GPR135◇ | A | Class A orphans | — | 1 | Tbio | 17 |
| GPR78 | GPR78◇ | A | Class A orphans | — | — | Tbio | 17 |
| TAS2R41 | TAS2R41 | T2 | Taste 2 receptors | — | 3 | Tclin | 17 |
| GPR162 | GPR162◇ | A | Class A orphans | — | — | Tbio | 16 |
| ADGRB3 | ADGRB3 | B2 | ADGRB | — | — | Tbio | 16 |
| GPR33 | GPR33◇ | A | Class A orphans | — | 1 | Tclin | 16 |
| GPR63 | GPR63◇ | A | Class A orphans | — | 3 | Tchem | 16 |
| GPR146 | GPR146◇ | A | Class A orphans | — | — | Tbio | 16 |
| GPR21 | GPR21◇ | A | Class A orphans | 5 | — | Tbio | 16 |
| ADGRB2 | ADGRB2 | B2 | ADGRB | — | — | Tbio | 16 |
| ADGRG5 | ADGRG5 | B2 | ADGRG | 1 | — | Tbio | 16 |
| GPR83 | GPR83◇ | A | Class A orphans | — | — | Tbio | 15 |
| ADGRF5 | ADGRF5 | B2 | ADGRF | — | — | Tbio | 15 |
| GPR85 | GPR85◇ | A | Class A orphans | — | — | Tbio | 15 |
| ADGRE1 | ADGRE1 | B2 | ADGRE | — | — | Tbio | 15 |
| GPR176 | GPR176◇ | A | Class A orphans | — | — | Tbio | 15 |
| GPR25 | GPR25◇ | A | Class A orphans | — | — | Tbio | 15 |
| GPR151 | GPR151◇ | A | Class A orphans | — | — | Tbio | 14 |
| ADGRA3 | ADGRA3 | B2 | ADGRA | — | — | Tbio | 14 |
| GPR173 | GPR173◇ | A | Class A orphans | — | — | Tbio | 14 |
| GPRC5C | GPRC5C◇ | C | Class C Orphans | — | — | Tbio | 14 |
| GPR107 | GPR107◇ | Other | Other GPCR orphans | — | — | Tbio | 14 |
| GPR31 | GPR31◇ | A | Class A orphans | — | — | Tbio | 14 |
| TAS2R60 | TAS2R60 | T2 | Taste 2 receptors | — | 3 | Tclin | 14 |
| ADGRG4 | ADGRG4 | B2 | ADGRG | 1 | — | Tbio | 14 |