Explorer
Tchem targets
120 receptors match — sorted by development interest.
Class
Development
System
Sort
| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| VIPR1 | VPAC₁ receptor | B1 | VIP and PACAP receptors | 3 | 100 | Tchem | 37 |
| GPR39 | GPR39◇ | A | Class A orphans | — | 166 | Tchem | 37 |
| GRM8 | mGlu₈ receptor | C | Metabotropic glutamate receptors | — | 293 | Tchem | 37 |
| P2RY14 | P2Y₁₄ receptor | A | P2Y receptors | — | 733 | Tchem | 37 |
| GPR174 | GPR174◇ | A | Class A orphans | 3 | 182 | Tchem | 37 |
| TAS1R3 | TAS1R3 | C | Taste 1 receptors | — | 377 | Tchem | 37 |
| LPAR3 | LPA₃ receptor | A | Lysophospholipid (LPA) receptors | — | 390 | Tchem | 37 |
| MCHR2 | MCH₂ receptor | A | Melanin-concentrating hormone | 1 | 257 | Tchem | 37 |
| RXFP4 | RXFP4 | A | Relaxin family peptide receptors | 3 | 144 | Tchem | 36 |
| PRLHR | PrRP receptor | A | Prolactin-releasing peptide receptors | 2 | 259 | Tchem | 36 |
| FFAR3 | FFA3 receptor | A | Free fatty acid receptors | 2 | 157 | Tchem | 35 |
| GPR4 | GPR4◇ | A | Class A orphans | — | 145 | Tchem | 35 |
| LPAR2 | LPA₂ receptor | A | Lysophospholipid (LPA) receptors | — | 397 | Tchem | 35 |
| LPAR6 | LPA₆ receptor | A | Lysophospholipid (LPA) receptors | — | 23 | Tchem | 35 |
| RXFP3 | RXFP3 | A | Relaxin family peptide receptors | — | 274 | Tchem | 35 |
| NPY4R | Y₄ receptor | A | Neuropeptide Y receptors | 1 | 543 | Tchem | 35 |
| GPR132 | GPR132◇ | A | Class A orphans | 4 | 71 | Tchem | 35 |
| QRFPR | QRFP receptor | A | Peptide P518 receptors | 2 | 254 | Tchem | 35 |
| CXCR6 | CXCR6 | A | Chemokine receptors | — | 114 | Tchem | 34 |
| RXFP2 | RXFP2 | A | Relaxin family peptide receptors | — | 29 | Tchem | 34 |
| NPBWR1 | NPBW1 receptor | A | Neuropeptide W/neuropeptide B receptors | — | 550 | Tchem | 34 |
| NPFFR2 | NPFF2 receptor | A | Neuropeptide FF/neuropeptide AF receptors | — | 409 | Tchem | 34 |
| TAS1R2 | TAS1R2 | C | Taste 1 receptors | — | 180 | Tchem | 34 |
| MRGPRX4 | MRGPRX4◇ | A | Class A orphans | 4 | 513 | Tchem | 34 |
| FZD1 | FZD₁ | F | Frizzled | 2 | 11 | Tchem | 34 |
| CCR10 | CCR10 | A | Chemokine receptors | — | 42 | Tchem | 33 |
| GPR3 | GPR3◇ | A | Class A orphans | 3 | 83 | Tchem | 33 |
| FZD2 | FZD₂ | F | Frizzled | — | 5 | Tchem | 33 |
| UTS2R | UT receptor | A | Urotensin receptors | — | 520 | Tchem | 32 |
| OXER1 | OXE receptor | A | Leukotriene receptors | — | 151 | Tchem | 32 |
| GPR34 | GPR34◇ | A | Class A orphans | 9 | 37 | Tchem | 32 |
| LPAR5 | LPA₅ receptor | A | Lysophospholipid (LPA) receptors | — | 316 | Tchem | 32 |
| LGR5 | LGR5◇ | A | Class A orphans | — | 5 | Tchem | 31 |
| GALR3 | GAL₃ receptor | A | Galanin receptors | — | 229 | Tchem | 31 |
| FZD5 | FZD₅ | F | Frizzled | 1 | 1 | Tchem | 31 |
| NPFFR1 | NPFF1 receptor | A | Neuropeptide FF/neuropeptide AF receptors | — | 187 | Tchem | 31 |
| GPR142 | GPR142◇ | A | Class A orphans | — | 409 | Tchem | 30 |
| XCR1 | XCR1 | A | Chemokine receptors | 1 | 3 | Tchem | 29 |
| P2RY10 | P2RY10◇ | A | Class A orphans | 1 | 122 | Tchem | 29 |
| LPAR4 | LPA₄ receptor | A | Lysophospholipid (LPA) receptors | — | 43 | Tchem | 28 |
| TAS1R1 | TAS1R1 | C | Taste 1 receptors | — | 200 | Tchem | 28 |
| MAS1 | MAS1◇ | A | Class A orphans | — | 11 | Tchem | 28 |
| GPR27 | GPR27◇ | A | Class A orphans | — | 114 | Tchem | 28 |
| LGR6 | LGR6◇ | A | Class A orphans | — | 8 | Tchem | 27 |
| GPR160 | GPR160◇ | A | Class A orphans | — | 58 | Tchem | 27 |
| GPR37 | GPR37◇ | A | Class A orphans | — | 2 | Tchem | 24 |
| GPR50 | GPR50◇ | A | Class A orphans | — | 1 | Tchem | 23 |
| ADGRG2 | ADGRG2 | B2 | ADGRG | — | 1 | Tchem | 23 |
| GPR15 | GPR15◇ | A | Class A orphans | 1 | 4 | Tchem | 23 |
| GPR61 | GPR61◇ | A | Class A orphans | 3 | 3 | Tchem | 22 |
| GPR75 | GPR75◇ | A | Class A orphans | — | 1 | Tchem | 22 |
| GPR87 | GPR87◇ | A | Class A orphans | — | 3 | Tchem | 22 |
| ACKR4 | ACKR4 | A | Chemokine receptors | — | 3 | Tchem | 21 |
| CMKLR2 | chemerin receptor 2 | A | Chemerin receptor | 2 | 18 | Tchem | 21 |
| GPR37L1 | GPR37L1◇ | A | Class A orphans | — | 2 | Tchem | 19 |
| GPR19 | GPR19◇ | A | Class A orphans | — | 1 | Tchem | 19 |
| ADGRL2 | ADGRL2 | B2 | ADGRL | — | 1 | Tchem | 18 |
| NPBWR2 | NPBW2 receptor | A | Neuropeptide W/neuropeptide B receptors | — | 5 | Tchem | 18 |
| GPR32 | GPR32◇ | A | Class A orphans | — | 4 | Tchem | 17 |
| GPR63 | GPR63◇ | A | Class A orphans | — | 3 | Tchem | 16 |
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