Explorer
Tclin targets
177 receptors match — sorted by development interest.
Class
Development
System
Sort
| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| PTGDR2 | DP₂ receptor | A | Prostanoid receptors | 6 | 921 | Tclin | 51 |
| MC2R | MC₂ receptor | A | Melanocortin receptors | 1 | 60 | Tclin | 50 |
| CXCR1 | CXCR1 | A | Chemokine receptors | 1 | 723 | Tclin | 50 |
| GPR183 | GPR183◇ | A | Class A orphans | 2 | 277 | Tclin | 49 |
| GPBAR1 | GPBA receptor | A | Bile acid receptors | 5 | 909 | Tclin | 49 |
| P2RY2 | P2Y₂ receptor | A | P2Y receptors | — | 723 | Tclin | 49 |
| GLP2R | GLP-2 receptor | B1 | Glucagon receptor family | 1 | 237 | Tclin | 48 |
| TAS2R14 | TAS2R14 | T2 | Taste 2 receptors | 15 | 328 | Tclin | 47 |
| C3AR1 | C3a receptor | A | Complement peptide receptors | 9 | 452 | Tclin | 47 |
| GPR17 | GPR17◇ | A | Class A orphans | 1 | 551 | Tclin | 47 |
| BDKRB1 | B₁ receptor | A | Bradykinin receptors | 1 | 927 | Tclin | 46 |
| P2RY6 | P2Y₆ receptor | A | P2Y receptors | — | 711 | Tclin | 45 |
| GHRHR | GHRH receptor | B1 | Glucagon receptor family | 3 | 8 | Tclin | 45 |
| GPR65 | GPR65◇ | A | Class A orphans | — | 139 | Tclin | 44 |
| FPR3 | FPR3 | A | Formylpeptide receptors | — | 812 | Tclin | 43 |
| SCTR | secretin receptor | B1 | Glucagon receptor family | 3 | 27 | Tclin | 42 |
| GPR68 | GPR68◇ | A | Class A orphans | — | 79 | Tclin | 41 |
| GPR18 | GPR18 | A | GPR18, GPR55 and GPR119 | — | 305 | Tclin | 41 |
| TAS2R38 | TAS2R38 | T2 | Taste 2 receptors | — | 22 | Tclin | 41 |
| P2RY4 | P2Y₄ receptor | A | P2Y receptors | — | 413 | Tclin | 39 |
| MRGPRX1 | MRGPRX1◇ | A | Class A orphans | 7 | 311 | Tclin | 38 |
| LTB4R2 | BLT₂ receptor | A | Leukotriene receptors | — | 498 | Tclin | 38 |
| NTSR2 | NTS₂ receptor | A | Neurotensin receptors | — | 361 | Tclin | 36 |
| ADGRF1 | ADGRF1 | B2 | ADGRF | 9 | 34 | Tclin | 36 |
| HCAR1 | HCA₁ receptor | A | Hydroxycarboxylic acid receptors | — | 385 | Tclin | 35 |
| GPR143 | GPR143◇ | Other | Other GPCR orphans | — | 2 | Tclin | 35 |
| GPRC5D | GPRC5D◇ | C | Class C Orphans | 2 | 1 | Tclin | 34 |
| P2RY11 | P2Y₁₁ receptor | A | P2Y receptors | — | 80 | Tclin | 34 |
| TAS2R46 | TAS2R46 | T2 | Taste 2 receptors | 3 | 39 | Tclin | 33 |
| TAS2R8 | TAS2R8 | T2 | Taste 2 receptors | — | 645 | Tclin | 32 |
| C5AR2 | C5a₂ receptor | A | Complement peptide receptors | — | 30 | Tclin | 32 |
| PTH2R | PTH2 receptor | B1 | Parathyroid hormone receptors | 1 | 25 | Tclin | 32 |
| P2RY13 | P2Y₁₃ receptor | A | P2Y receptors | — | 35 | Tclin | 31 |
| TAS2R1 | TAS2R1 | T2 | Taste 2 receptors | — | 10 | Tclin | 31 |
| TAS2R16 | TAS2R16 | T2 | Taste 2 receptors | — | 15 | Tclin | 29 |
| FZD8 | FZD₈ | F | Frizzled | — | 2 | Tclin | 27 |
| TAS2R43 | TAS2R43 | T2 | Taste 2 receptors | — | 15 | Tclin | 24 |
| TAS2R4 | TAS2R4 | T2 | Taste 2 receptors | — | 8 | Tclin | 24 |
| TAS2R31 | TAS2R31 | T2 | Taste 2 receptors | — | 25 | Tclin | 23 |
| TAS2R39 | TAS2R39 | T2 | Taste 2 receptors | — | 17 | Tclin | 23 |
| TAS2R10 | TAS2R10 | T2 | Taste 2 receptors | — | 13 | Tclin | 22 |
| TAS2R20 | TAS2R20 | T2 | Taste 2 receptors | — | 7 | Tclin | 22 |
| ADGRG3 | ADGRG3 | B2 | ADGRG | 2 | 1 | Tclin | 21 |
| TAS2R50 | TAS2R50 | T2 | Taste 2 receptors | — | 3 | Tclin | 21 |
| TAS2R9 | TAS2R9 | T2 | Taste 2 receptors | — | 6 | Tclin | 21 |
| TAS2R5 | TAS2R5 | T2 | Taste 2 receptors | — | 4 | Tclin | 19 |
| TAS2R7 | TAS2R7 | T2 | Taste 2 receptors | — | 4 | Tclin | 19 |
| TAS2R13 | TAS2R13 | T2 | Taste 2 receptors | — | 4 | Tclin | 18 |
| TAS2R19 | TAS2R19 | T2 | Taste 2 receptors | — | 1 | Tclin | 18 |
| TAS2R3 | TAS2R3 | T2 | Taste 2 receptors | — | 2 | Tclin | 18 |
| TAS2R40 | TAS2R40 | T2 | Taste 2 receptors | — | 5 | Tclin | 18 |
| TAS2R42 | TAS2R42 | T2 | Taste 2 receptors | — | 1 | Tclin | 17 |
| TAS2R41 | TAS2R41 | T2 | Taste 2 receptors | — | 3 | Tclin | 17 |
| GPR33 | GPR33◇ | A | Class A orphans | — | 1 | Tclin | 16 |
| TAS2R60 | TAS2R60 | T2 | Taste 2 receptors | — | 3 | Tclin | 14 |
| TAS2R30 | TAS2R30 | T2 | Taste 2 receptors | — | 4 | Tclin | 13 |
| TAS2R45 | TAS2R45 | T2 | Taste 2 receptors | — | 1 | Tclin | 9 |
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