Explorer
Tbio targets
97 receptors match — sorted by development interest.
Class
Development
System
Sort
| Gene | Receptor | Class | Family | Structures | Ligands | TDL | Dev. interest |
|---|---|---|---|---|---|---|---|
| RHO | Rhodopsin | A | Opsins | 4 | — | Tbio | 50 |
| FZD6 | FZD₆ | F | Frizzled | 2 | 4 | Tbio | 36 |
| CRHR1 | CRF₁ receptor | B1 | Corticotropin-releasing factor receptors | 7 | — | Tbio | 35 |
| ADGRG1 | ADGRG1 | B2 | ADGRG | 1 | — | Tbio | 30 |
| OXGR1 | oxoglutarate receptor | A | Oxoglutarate receptors | — | 12 | Tbio | 28 |
| GPR161 | GPR161◇ | A | Class A orphans | 2 | — | Tbio | 27 |
| CELSR1 | CELSR1 | B2 | ADGRC | — | — | Tbio | 27 |
| ADGRV1 | ADGRV1 | B2 | ADGRV | — | — | Tbio | 26 |
| GPR101 | GPR101◇ | A | Class A orphans | 3 | — | Tbio | 26 |
| GPRC6A | GPRC6 receptor◇ | C | Class C Orphans | — | 8 | Tbio | 26 |
| OPN1LW | OPN1LW | A | Opsins | 1 | — | Tbio | 25 |
| FZD3 | FZD₃ | F | Frizzled | 3 | — | Tbio | 25 |
| GPR179 | GPR179◇ | C | Class C Orphans | 1 | — | Tbio | 25 |
| ADGRG6 | ADGRG6 | B2 | ADGRG | — | — | Tbio | 24 |
| GPR158 | GPR158◇ | C | Class C Orphans | 5 | — | Tbio | 24 |
| OPN1MW | OPN1MW | A | Opsins | — | — | Tbio | 24 |
| F2RL2 | PAR3 | A | Proteinase-activated receptors | — | — | Tbio | 24 |
| GPR12 | GPR12◇ | A | Class A orphans | 1 | 2 | Tbio | 24 |
| ACKR1 | ACKR1 | A | Chemokine receptors | 1 | — | Tbio | 24 |
| CELSR2 | CELSR2 | B2 | ADGRC | — | — | Tbio | 24 |
| ACKR2 | ACKR2 | A | Chemokine receptors | — | 6 | Tbio | 23 |
| OPN1SW | OPN1SW | A | Opsins | — | — | Tbio | 23 |
| ADGRL3 | ADGRL3 | B2 | ADGRL | 2 | — | Tbio | 23 |
| P2RY8 | P2RY8◇ | A | Class A orphans | — | — | Tbio | 23 |
| ADGRD1 | ADGRD1 | B2 | ADGRD | 2 | — | Tbio | 23 |
| ADGRE5 | ADGRE5 | B2 | ADGRE | 6 | 2 | Tbio | 23 |
| MRGPRD | MRGPRD◇ | A | Class A orphans | 6 | 1 | Tbio | 22 |
| ADGRL1 | ADGRL1 | B2 | ADGRL | — | — | Tbio | 22 |
| GPR156 | GPR156◇ | C | Class C Orphans | 5 | — | Tbio | 22 |
| OPN4 | OPN4 | A | Opsins | — | — | Tbio | 21 |
| TAAR5 | TAAR5◇ | A | Class A orphans | — | 2 | Tbio | 21 |
| RRH | RRH | A | Opsins | — | — | Tbio | 21 |
| GPR20 | GPR20◇ | A | Class A orphans | 3 | — | Tbio | 20 |
| GPRC5A | GPRC5A◇ | C | Class C Orphans | — | — | Tbio | 20 |
| ADGRE2 | ADGRE2 | B2 | ADGRE | — | — | Tbio | 20 |
| GPRC5B | GPRC5B◇ | C | Class C Orphans | — | — | Tbio | 20 |
| GPR137 | GPR137◇ | Other | Other GPCR orphans | — | — | Tbio | 19 |
| CELSR3 | CELSR3 | B2 | ADGRC | — | — | Tbio | 19 |
| FZD10 | FZD₁₀ | F | Frizzled | — | — | Tbio | 18 |
| OPN5 | OPN5 | A | Opsins | — | — | Tbio | 18 |
| ADGRL4 | ADGRL4 | B2 | ADGRL | — | — | Tbio | 18 |
| GPR26 | GPR26◇ | A | Class A orphans | — | — | Tbio | 18 |
| OPN3 | OPN3 | A | Opsins | — | — | Tbio | 17 |
| ADGRB1 | ADGRB1 | B2 | ADGRB | — | 1 | Tbio | 17 |
| GPR135 | GPR135◇ | A | Class A orphans | — | 1 | Tbio | 17 |
| GPR78 | GPR78◇ | A | Class A orphans | — | — | Tbio | 17 |
| GPR162 | GPR162◇ | A | Class A orphans | — | — | Tbio | 16 |
| ADGRB3 | ADGRB3 | B2 | ADGRB | — | — | Tbio | 16 |
| GPR146 | GPR146◇ | A | Class A orphans | — | — | Tbio | 16 |
| GPR21 | GPR21◇ | A | Class A orphans | 5 | — | Tbio | 16 |
| ADGRB2 | ADGRB2 | B2 | ADGRB | — | — | Tbio | 16 |
| ADGRG5 | ADGRG5 | B2 | ADGRG | 1 | — | Tbio | 16 |
| GPR83 | GPR83◇ | A | Class A orphans | — | — | Tbio | 15 |
| ADGRF5 | ADGRF5 | B2 | ADGRF | — | — | Tbio | 15 |
| GPR85 | GPR85◇ | A | Class A orphans | — | — | Tbio | 15 |
| ADGRE1 | ADGRE1 | B2 | ADGRE | — | — | Tbio | 15 |
| GPR176 | GPR176◇ | A | Class A orphans | — | — | Tbio | 15 |
| GPR25 | GPR25◇ | A | Class A orphans | — | — | Tbio | 15 |
| GPR151 | GPR151◇ | A | Class A orphans | — | — | Tbio | 14 |
| ADGRA3 | ADGRA3 | B2 | ADGRA | — | — | Tbio | 14 |
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